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Cat. No. Product Name Target Signaling Pathways
T11626 IACS-8968

IDO/TDO Inhibitor

IDO Metabolism
IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).
T11627 IACS-8968 R-enantiomer

IDO/TDO Inhibitor (R-enantiomer)

IDO Metabolism
IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).
T11628 IACS-8968 S-enantiomer

IDO/TDO Inhibitor (S-enantiomer)

IDO Metabolism
IACS-8968 S-enantiomer is the S-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).
T4410 LM10

Others Others
LM10 是有效的色氨酸 2,3-双加氧酶的抑制剂。色氨酸 2,3-双加氧酶是一种无关的肝酶,它可通过犬尿氨酸途径降解色氨酸。它对研究癌症疾病具有潜在的研究价值。
T11623 IDO/TDO-IN-1

Others Others
IDO/TDO-IN-1 is an orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50s: 9.7 and 47 nM).
T74536 IDO/Tubulin-IN-2

IDO/Tubulin-IN-2 (HT2) 是一种对TDO和微管蛋白 (tubulin)展现出高效抑制作用的化合物。该抑制剂对多种癌细胞系(包括U87、HepG2、A549、HCT-116和LO2)均表现出强抗肿瘤活性,其半抑制浓度(IC50)分别为0.43、0.036、0.041、0.095和1.04 μM,有效提升了抗肿瘤效果。

化合物

IACS-8968
Cat.No: T11626
Synonym: IDO/TDO Inhibitor
Target: IDO
IACS-8968 R-enantiomer
Cat.No: T11627
Synonym: IDO/TDO Inhibitor (R-enantiomer)
Target: IDO
IACS-8968 S-enantiomer
Cat.No: T11628
Synonym: IDO/TDO Inhibitor (S-enantiomer)
Target: IDO
LM10
Cat.No: T4410
Synonym:
Target: Others
IDO/TDO-IN-1
Cat.No: T11623
Synonym:
Target: Others
IDO/Tubulin-IN-2
Cat.No: T74536
Synonym:
Target:
TargetMol Loading
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